SCHEMBL4307660

SCHEMBL4307660

CC(C)(C)OC(=O)N[C@H](C(=O)N1C[C@H](OCc2cccc(-c3cccc(Br)c3)c2)C[C@H]1C(=O)O)C1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.40
ACE P12821 1/20 0.40
CTSB P07858 2/20 0.39
CTSS P25774 2/20 0.39
CTSK P43235 2/20 0.39
CTSL P07711 1/20 0.39
AAK1 Q2M2I8 3/20 0.38
AGTR2 P50052 2/20 0.38
REN P00797 2/20 0.37
CMA1 P23946 1/20 0.37
ABCB1 P08183 1/20 0.37
USP30 Q70CQ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2430508 0.93 CACNA1B (0.41) CACNA1BACECTSBCTSSCTSK
SCHEMBL4294862 0.89 ACE (0.40) CACNA1BACECTSBCTSSCTSK
SCHEMBL2426240 0.83 KLK5 (0.40) CACNA1BACECTSBCTSSCTSK
SCHEMBL2430509 0.82 CACNA1B (0.39) CACNA1BCTSBCTSSCTSKCTSL
SCHEMBL4301232 0.78 NAAA (0.44) AGTR2
SCHEMBL8227117 0.76 USP30 (0.43) ABCB1USP30
SCHEMBL2744335 0.76 AAK1 (0.40) CACNA1BACECTSLAAK1
SCHEMBL6745052 0.74 CMA1 (0.53) AGTR2CMA1ABCB1
SCHEMBL4303372 0.72 AGTR2 (0.36) AGTR2ABCB1
SCHEMBL2426243 0.72 CTSL (0.38) CACNA1BACECTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8314062-B2 Macrocyclic compounds as antiviral agents INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2012-11-20 US disclosed
US-20090312241-A1 Macrocyclic Compounds as Antiviral Agents ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2009-12-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312241-A1 Macrocyclic Compounds as Antiviral Agents ZC3HAV1, ZC3HAV1L, HAVCR2 CACNA1B 3771/4885ACE 204/4885CTSB 476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.