SCHEMBL24282005

SCHEMBL24282005

COC(=O)c1ccc2nc(F)[nH]c2c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.68
LMNA P02545 4/20 0.68
KDM4E B2RXH2 3/20 0.68
ALDH1A1 P00352 3/20 0.68
L3MBTL1 Q9Y468 1/20 0.68
BRD4 O60885 1/20 0.54
MMP2 P08253 1/20 0.53
MMP9 P14780 1/20 0.53
MMP8 P22894 1/20 0.53
MMP13 P45452 1/20 0.53
KDR P35968 2/20 0.51
MAPK1 P28482 2/20 0.51
ADORA3 P0DMS8 1/20 0.51
PTGS1 P23219 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
IRAK4 Q9NWZ3 1/20 0.49
PARP1 P09874 2/20 0.49
KIF11 P52732 1/20 0.49
ALOX15 P16050 1/20 0.49
RHEB Q15382 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682076 0.85 ALDH1A1 (0.64) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL4243540 0.83 HSP90AA1 (0.69) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL6217370 0.82 HTT (0.64) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL1097139 0.82 HTT (0.64) HTTLMNAKDM4EALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL7324046 0.82 HSP90AA1 (0.68) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL28396605 0.82 HTT (0.64) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL30349840 0.81 ALDH1A1 (0.64) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL6088752 0.81 ALDH1A1 (1.00) HTTLMNAKDM4EALDH1A1L3MBTL1
SCHEMBL27978054 0.81 TDP1 (0.66) ALDH1A1MMP2MMP9MMP8MMP13
SCHEMBL20982471 0.81 MMP2 (0.78) HTTLMNAKDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022074617-A1 COMBINATION OF ANTIBODY-DRUG CONJUGATE AND PARP1 SELECTIVE INHIBITOR ASTRAZENECA UK LIMITED (GB) 2022-04-14 WO disclosed