SCHEMBL24282902

SCHEMBL24282902

CC(C)(C)OC(=O)N[C@H]1CC(=O)N(c2ccc3c(cnn3-c3ccc(F)cc3)c2)[C@@H]1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.46
NR3C1 P04150 14/20 0.46
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.42
PGR P06401 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21104148 0.93 NR3C1 (0.44) SMONR3C1MAPK1PGR
SCHEMBL21057716 0.90 SMO (0.49) SMONR3C1PGR
SCHEMBL21058104 0.89 SMO (0.50) SMONR3C1MAPK1PGR
SCHEMBL21058051 0.85 SMO (0.45) SMONR3C1MAPK1
SCHEMBL21057753 0.85 SMO (0.45) SMONR3C1MAPK1
SCHEMBL21057805 0.85 SMO (0.45) SMONR3C1MAPK1
SCHEMBL29525941 0.85 SMO (0.45) SMONR3C1MAPK1
SCHEMBL28448055 0.81 SMO (0.47) SMONR3C1MAPK1PGR
SCHEMBL21057922 0.80 NR3C1 (0.48) SMONR3C1MAPK1PGR
SCHEMBL21057722 0.79 SMO (0.49) SMONR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12344605-B2 Substituted pyrrolidine amides II GRUENENTHAL GMBH (DE) 2025-07-01 US disclosed
US-20220127264-A1 SUBSTITUTED PYRROLIDINE AMIDES II GRUENENTHAL GMBH (DE) 2022-04-28 US disclosed
US-20220127264-A1 SUBSTITUTED PYRROLIDINE AMIDES II GRUENENTHAL GMBH (DE) 2022-04-28 US disclosed
EP-3728233-B1 SUBSTITUTED PYRROLIDINE AMIDES II GRUENENTHAL GMBH (DE) 2022-04-20 EP disclosed
EP-3728233-B1 SUBSTITUTED PYRROLIDINE AMIDES II GRUENENTHAL GMBH (DE) 2022-04-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220127264-A1 SUBSTITUTED PYRROLIDINE AMIDES II NR3C1, NR3C2, MC2R SMO 4592/4885NR3C1 1/4885TP53 3674/4885
US-12344605-B2 Substituted pyrrolidine amides II NR3C1, NR3C2, MC2R SMO 4592/4885NR3C1 1/4885TP53 3674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.