SCHEMBL24286262

SCHEMBL24286262

O=C1COc2cc(Cl)c(Br)cc2N1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.49
PARP1 P09874 1/20 0.45
MAPT P10636 7/20 0.44
ALDH1A1 P00352 2/20 0.44
TP53 P04637 5/20 0.44
THRB P10828 1/20 0.44
PKM P14618 2/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
AHR P35869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18264334 0.93 MMP12 (0.49) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL30015636 0.93 MMP12 (0.49) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL2945700 0.86 MMP12 (0.54) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL2955843 0.86 MMP12 (0.54) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL18152757 0.80 MMP12 (0.49) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL3342717 0.80 MMP12 (0.49) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL8192799 0.80 NR3C2 (0.51) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL3592276 0.80 MMP12 (0.49) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL21552385 0.80 MMP12 (0.49) MMP12PARP1MAPTALDH1A1TP53
SCHEMBL305188 0.80 MMP12 (0.57) MMP12PARP1MAPTALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3307738-B1 ARYL DIHYDRO-2H-BENZO[B][1,4]OXAZINE SULFONAMIDE AND RELATED COMPOUNDS FOR USE AS AGONISTS OF RORY AND THE TREATMENT OF DISEASE UNIV MICHIGAN REGENTS (US) 2022-04-20 EP disclosed