SCHEMBL24286751

SCHEMBL24286751

Fc1ccc(-c2ccc3c(c2)NCCC3)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.48
PYGL P06737 1/20 0.41
HRH3 Q9Y5N1 2/20 0.41
PARP10 Q53GL7 2/20 0.39
PARP1 P09874 1/20 0.39
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
DHFR P00374 1/20 0.38
TTR P02766 1/20 0.38
ALB P02768 1/20 0.38
HMGB1 P09429 1/20 0.38
HPGD P15428 1/20 0.38
CXCL12 P48061 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24286750 0.88 PARP10 (0.42) TDP2PYGLHRH3PARP10PARP1
SCHEMBL24286723 0.86 PYGL (0.50) TDP2PYGLHRH3PARP10PARP1
SCHEMBL24287001 0.84 PARP1 (0.44) PYGLHRH3PARP1KDM4EALDH1A1
SCHEMBL3112268 0.82 PYGL (0.49) PYGLHRH3PARP10PARP1KDM4E
SCHEMBL29622425 0.82 PYGL (0.49) PYGLHRH3PARP10PARP1KDM4E
SCHEMBL24287059 0.82 PYGL (0.39) TDP2PYGLHRH3PARP10PARP1
Hydrochloric Acid SCHEMBL30142485 0.81 PYGL (0.48) PYGLHRH3PARP10PARP1KDM4E
Hydrochloric Acid SCHEMBL2144161 0.81 PYGL (0.48) PYGLHRH3PARP10PARP1KDM4E
SCHEMBL24287074 0.79 PARP10 (0.50) PYGLHRH3PARP10KDM4EMEN1
SCHEMBL24287049 0.78 PGR (0.41) PYGLHRH3PARP10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3307738-B1 ARYL DIHYDRO-2H-BENZO[B][1,4]OXAZINE SULFONAMIDE AND RELATED COMPOUNDS FOR USE AS AGONISTS OF RORY AND THE TREATMENT OF DISEASE UNIV MICHIGAN REGENTS (US) 2022-04-20 EP disclosed