SCHEMBL24310644

SCHEMBL24310644

CCCC(=O)c1ncn(Cc2ccc(OC(F)(F)F)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
TSHR P16473 1/20 0.45
CACNA1H O95180 3/20 0.43
CACNA1G O43497 2/20 0.43
CACNA1I Q9P0X4 2/20 0.43
ALDH1A1 P00352 5/20 0.42
HPGD P15428 4/20 0.41
KDM4E B2RXH2 3/20 0.41
KLKB1 P03952 1/20 0.41
KLK1 P06870 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
GAA P10253 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
AADAT Q8N5Z0 1/20 0.40
CYP2C9 P11712 3/20 0.40
CYP2C19 P33261 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24310654 0.85 HDAC1 (0.43) HDAC1HDAC6CACNA1HCACNA1GCACNA1I
SCHEMBL22737100 0.84 HDAC1 (0.50) HDAC1HDAC6TSHRCACNA1HCACNA1G
SCHEMBL24310340 0.83 HDAC1 (0.48) HDAC1HDAC6ALDH1A1HPGDTP53
SCHEMBL20095692 0.80 KLKB1 (0.47) HDAC1HDAC6ALDH1A1KLKB1KLK1
SCHEMBL8532976 0.77 KLKB1 (0.53) TSHRCACNA1HCACNA1GCACNA1IKLKB1
SCHEMBL24310730 0.74 HDAC1 (0.45) HDAC1HDAC6CACNA1HCACNA1GCACNA1I
SCHEMBL22737096 0.73 CACNA1H (0.46) HDAC1HDAC6TSHRCACNA1HCACNA1G
SCHEMBL28517031 0.73 HDAC1 (0.45) HDAC1HDAC6TSHRCACNA1HCACNA1G
SCHEMBL8531702 0.72 CACNA1H (0.55) TSHRCACNA1HCACNA1GCACNA1IALDH1A1
SCHEMBL24310660 0.72 GLA (0.48) HDAC1HDAC6CACNA1HCACNA1GCACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3978492-A1 BICYCLIC COMPOUND AS RIP-1 KINASE INHIBITOR AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2022-04-06 EP disclosed