SCHEMBL28517031

SCHEMBL28517031

CNc1ncn(Cc2ccc(OC(F)(F)F)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
CACNA1H O95180 3/20 0.43
CACNA1G O43497 2/20 0.43
CACNA1I Q9P0X4 2/20 0.43
GPR39 O43194 1/20 0.42
AADAT Q8N5Z0 1/20 0.39
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
CHRNA7 P36544 1/20 0.38
TEAD1 P28347 1/20 0.38
VNN1 O95497 1/20 0.38
EPHX2 P34913 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
BRD4 O60885 1/20 0.38
MBOAT4 Q96T53 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22737100 0.78 HDAC1 (0.50) HDAC1HDAC6ALDH1A1TSHRCACNA1H
SCHEMBL21492990 0.77 HDAC1 (0.43) HDAC1HDAC6ALDH1A1TSHRCACNA1H
SCHEMBL17132895 0.76 ALDH1A1 (0.48) HDAC1HDAC6ALDH1A1HTR2CSLC6A4
SCHEMBL22737096 0.76 CACNA1H (0.46) HDAC1HDAC6ALDH1A1TSHRCACNA1H
SCHEMBL31272703 0.73 MAPT (0.38) HDAC1HDAC6ALDH1A1CACNA1HCACNA1G
SCHEMBL24310644 0.73 HDAC1 (0.45) HDAC1HDAC6ALDH1A1TSHRCACNA1H
Hydrochloric Acid SCHEMBL28525601 0.72 KLKB1 (0.46) ALDH1A1TSHRCACNA1HCACNA1GCACNA1I
SCHEMBL3319305 0.71 CYP19A1 (0.57) HDAC1HDAC6ALDH1A1TSHRCACNA1H
SCHEMBL28530827 0.70 CACNA1G (0.43) HDAC1HDAC6TSHRCACNA1HCACNA1G
SCHEMBL8641487 0.69 CACNA1H (0.52) HDAC1HDAC6ALDH1A1TSHRCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-A Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2021-01-12 CN disclosed