SCHEMBL24313748

SCHEMBL24313748

O=Cc1c(O)cc(C2CC2)cc1-n1ccnc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.40
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
CHRNA7 P36544 1/20 0.34
EGLN2 Q96KS0 1/20 0.33
ENPP2 Q13822 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
CD38 P28907 3/20 0.32
CYP17A1 P05093 1/20 0.30
CYP21A2 P08686 1/20 0.30
CYP11B1 P15538 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29588780 1.00 IDO1 (0.40) IDO1HTR2AHTR2CHTR2BCHRNA7
SCHEMBL24313632 0.81 CYP11B1 (0.43) CYP11B1
SCHEMBL12174452 0.69 HDAC4 (0.42)
SCHEMBL24313611 0.67 ESR2 (0.36)
SCHEMBL24313736 0.67 TBXAS1 (0.39) HTR2AHTR2CHTR2BCA12CA9
SCHEMBL29588188 0.67 TBXAS1 (0.39) HTR2AHTR2CHTR2BCA12CA9
SCHEMBL31005858 0.67 CD38 (0.41) HTR2AHTR2CHTR2BCD38
SCHEMBL25192493 0.67 CD38 (0.41) HTR2AHTR2CHTR2BCD38
SCHEMBL24313735 0.64 HTR2A (0.35) HTR2AHTR2CHTR2B
SCHEMBL24314202 0.64 ESR2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022081842-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed