SCHEMBL2431412

SCHEMBL2431412

C[Si](C)(C)C#Cc1nccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
PLAU P00749 2/20 0.44
F12 P00748 1/20 0.44
NCF1 P14598 1/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
BACE1 P56817 1/20 0.44
PLG P00747 1/20 0.41
CYP3A4 P08684 3/20 0.38
HRH4 Q9H3N8 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 3/20 0.37
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15947640 0.85 PLAU (0.54) CYP2A6PLAUF12NCF1NOS3
SCHEMBL29937111 0.81 CYP2A6 (0.44) CYP2A6PLAUF12NCF1NOS3
SCHEMBL3790627 0.77 GRM5 (0.51) CYP2A6PLAUF12NCF1NOS3
SCHEMBL15940603 0.76 ADORA2A (0.54) CYP2A6PLAUF12NCF1NOS3
Hydrochloric Acid SCHEMBL8116929 0.75 ADORA2A (0.53) CYP2A6PLAUF12NCF1NOS3
SCHEMBL17370957 0.75 CHAT (0.49) CYP2A6PLAUF12NCF1NOS3
SCHEMBL15947643 0.75 CYP2A6 (0.49) CYP2A6PLAUF12NCF1NOS3
SCHEMBL194554 0.73 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL2852412 0.73 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL2418686 0.73 CYP2A6 (0.50) CYP2A6PLAUF12NCF1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2542239-A1 USE OF ISOQUINOLONES FOR PREPARING DRUGS, NOVEL ISOQUINOLONES AND METHOD FOR SYNTHESISING SAME Université Joseph Fourier (FR) 2013-01-09 EP disclosed
WO-2011107709-A1 USE OF ISOQUINOLONES FOR PREPARING DRUGS, NOVEL ISOQUINOLONES AND METHOD FOR SYNTHESISING SAME UNIVERSITE JOSEPH FOURIER (FR) 2011-09-09 WO disclosed