SCHEMBL2418686

SCHEMBL2418686

C#Cc1nccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.50
PLAU P00749 2/20 0.50
F12 P00748 1/20 0.50
NCF1 P14598 1/20 0.50
NOS3 P29474 1/20 0.50
NOS1 P29475 1/20 0.50
NOS2 P35228 1/20 0.50
BACE1 P56817 1/20 0.50
PLG P00747 1/20 0.42
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 2/20 0.41
ALDH1A1 P00352 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CFTR P13569 1/20 0.41
GOPC Q9HD26 1/20 0.41
CYP3A4 P08684 3/20 0.40
APEX1 P27695 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15947640 0.83 PLAU (0.54) CYP2A6PLAUF12NCF1NOS3
SCHEMBL29358794 0.79 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL251028 0.79 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL194554 0.79 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL2852412 0.79 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL7544045 0.79 PLAU (0.50) CYP2A6PLAUF12NCF1NOS3
SCHEMBL27933452 0.76 KDM4E (0.45) MAPTLMNANPC1ALDH1A1RAB9A
SCHEMBL15940603 0.75 ADORA2A (0.54) CYP2A6PLAUF12NCF1NOS3
Hydrochloric Acid SCHEMBL8116929 0.73 ADORA2A (0.53) CYP2A6PLAUF12NCF1NOS3
SCHEMBL2431412 0.73 CYP2A6 (0.48) CYP2A6PLAUF12NCF1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11005050-B2 Metal complexes MERCK PATENT GMBH (DE) 2021-05-11 US disclosed
CN-106661031-B Pyrrolopyrimidine compounds or its salt, pharmaceutical composition and application containing it 大鹏药品工业株式会社 2019-07-23 CN disclosed
US-20190010158-A1 ANTITUMOR EFFECT POTENTIATOR COMPRISING PYRROLOPYRIMIDINE COMPOUND TAIHO PHARMACETUICAL CO., LTD. (JP) 2019-01-10 US disclosed
US-10174040-B2 Pyrrolopyrimidine compound or salt thereof and compositions containing the pyrrolopyrimidine compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2019-01-08 US disclosed
EP-3395345-A1 ANTITUMOR EFFECT POTENTIATOR COMPRISING PYRROLOPYRIMIDINE COMPOUND Taiho Pharmaceutical Co., Ltd. (JP) 2018-10-31 EP disclosed
EP-3102650-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2018-08-29 EP disclosed
US-20180162864-A1 PYRROLOPYRIMIDINE COMPOUND OR SALT THEREOF AND COMPOSITIONS CONTAINING THE PYRROLOPYRIMIDINE COMPOUND OR SALT THEREOF TAIHO PHARMACEUTICAL CO., LTD. (JP) 2018-06-14 US disclosed
US-9963456-B2 Pyrrolopyrimidine compound or salt thereof and compositions containing the pyrrolopyrimidine compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD (JP) 2018-05-08 US disclosed
EP-3094638-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-11-08 EP disclosed
EP-3094638-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-11-08 EP disclosed
WO-2015117718-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2015-08-13 WO disclosed
WO-2015104045-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2015-07-16 WO disclosed
US-8723017-B2 Dye sensitised solar cell BASF SE (DE) 2014-05-13 US disclosed
EP-2553698-A1 DYE SENSITISED SOLAR CELL BASF SE (DE) 2013-02-06 EP disclosed
EP-2253031-B1 DYE SENSITISED SOLAR CELL BASF SE (DE) 2012-10-17 EP disclosed
WO-2011120908-A1 DYE SENSITISED SOLAR CELL BASF SE (DE) 2011-10-06 WO disclosed
US-20110233477-A1 Dye sensitised solar cell BASF SE (DE) 2011-09-29 US disclosed
US-20110061723-A1 DYE SENSITISED SOLAR CELL BASF SE (DE) 2011-03-17 US disclosed
EP-2253031-A1 DYE SENSITISED SOLAR CELL BASF SE (DE) 2010-11-24 EP disclosed
WO-2009109499-A1 DYE SENSITISED SOLAR CELL BASF SE (DE) 2009-09-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190010158-A1 ANTITUMOR EFFECT POTENTIATOR COMPRISING PYRROLOPYRIMIDINE COMPOUND MCL1, TP53, DPYD CYP2A6 4389/4885PLAU 1796/4885F12 4883/4885
US-20110233477-A1 Dye sensitised solar cell SLC11A2, CRY1, MPO CYP2A6 2926/4885PLAU 4354/4885F12 3702/4885
US-10174040-B2 Pyrrolopyrimidine compound or salt thereof and compositions containing the pyrrolopyrimidine compound or salt thereof KRAS, DPYD, PSTPIP2 CYP2A6 3788/4885PLAU 3050/4885F12 4463/4885
US-20110061723-A1 DYE SENSITISED SOLAR CELL FTO, TET1, METTL14 CYP2A6 3489/4885PLAU 4090/4885F12 4551/4885
US-11005050-B2 Metal complexes SOD1, AP1M1, AP3M1 CYP2A6 3927/4885PLAU 2801/4885F12 2850/4885
US-20180162864-A1 PYRROLOPYRIMIDINE COMPOUND OR SALT THEREOF AND COMPOSITIONS CONTAINING THE PYRROLOPYRIMIDINE COMPOUND OR SALT THEREOF KRAS, DPYD, PSTPIP2 CYP2A6 3788/4885PLAU 3050/4885F12 4463/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.