SCHEMBL24314237

SCHEMBL24314237

CCOc1ccc(F)cc1S(=O)(=O)NC(=O)c1cc2c(F)cc(C3CC3)cc2o1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 7/20 0.38
TSPO P30536 2/20 0.38
ALPL P05186 5/20 0.37
KAT6A Q92794 2/20 0.37
MCHR1 Q99705 2/20 0.36
KCNH2 Q12809 1/20 0.36
HRH1 P35367 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24314247 0.94 MEN1 (0.36) MRGPRX1TSPOKAT6AMEN1KMT2A
SCHEMBL24313659 0.93 MRGPRX1 (0.36) MRGPRX1TSPOKAT6AMCHR1KCNH2
SCHEMBL24313753 0.92 MEN1 (0.38) MRGPRX1TSPOKAT6AMEN1KMT2A
SCHEMBL24313760 0.90 SCN9A (0.35) MEN1KMT2AL3MBTL1TSHR
SCHEMBL24313686 0.90 ALDH1A1 (0.44) ALPLMCHR1KCNH2MEN1KMT2A
SCHEMBL24314300 0.90 ALDH1A1 (0.38) MRGPRX1TSPOALPLMCHR1KCNH2
SCHEMBL24313979 0.90 CYP1A2 (0.37) ALPLMCHR1KCNH2MEN1KMT2A
SCHEMBL24314309 0.88 SCN7A (0.37) ALPLMCHR1MEN1KMT2AL3MBTL1
SCHEMBL24314230 0.88 MEN1 (0.36) KAT6AMEN1KMT2A
SCHEMBL24313965 0.85 LMNA (0.38) MRGPRX1KAT6AMCHR1KCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4229045-B1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER BROAD INST INC (US) 2025-11-12 EP claimed
EP-4229045-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER The Broad Institute Inc. (US) 2023-08-23 EP claimed
WO-2022081842-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO claimed
EP-4229045-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER The Broad Institute Inc. (US) 2023-08-23 EP disclosed
WO-2022081842-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed
WO-2022081842-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed