SCHEMBL24316039

SCHEMBL24316039

Fc1ccc2c(c1)CCCN2I

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PDK3 Q15120 1/20 0.46
PDK4 Q16654 1/20 0.46
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
ROCK1 Q13464 1/20 0.40
ALDH1A1 P00352 4/20 0.39
GAA P10253 2/20 0.39
HTT P42858 1/20 0.39
CNR2 P34972 1/20 0.38
TRPA1 O75762 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4C Q9H3R0 1/20 0.37
NR1I2 O75469 1/20 0.36
RORC P51449 1/20 0.36
NR1H2 P55055 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2625790 0.78 ALDH1A1 (0.58) NOTUMHDAC1HDAC6PDK1PDK2
SCHEMBL20427833 0.78 ALDH1A1 (0.58) NOTUMPDK1PDK2PDK3PDK4
SCHEMBL7257879 0.78 NOTUM (0.46) NOTUMHDAC1HDAC6PDK1PDK2
SCHEMBL23346736 0.78 PDK1 (0.46) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL16511459 0.74 ALDH1A1 (0.50) HDAC1HDAC6HTR2CHTR2BALDH1A1
SCHEMBL21524785 0.74 HSD17B10 (0.58) NOTUMPDK1PDK2PDK3PDK4
SCHEMBL8728886 0.74 HDAC1 (0.52) NOTUMHDAC1HDAC6PDK1PDK2
SCHEMBL24824408 0.74 NOTUM (0.46) NOTUMHDAC1HDAC6PDK1PDK2
SCHEMBL12382109 0.74 NOTUM (0.46) NOTUMHDAC1HDAC6PDK1PDK2
SCHEMBL7733872 0.74 ALDH1A1 (0.67) NOTUMHDAC1HDAC6PDK1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022081925-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 C4 THERAPEUTICS, INC. (US) 2022-04-21 WO disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed