SCHEMBL24317548

SCHEMBL24317548

CCc1nnc(-c2nnc(CC)[nH]2)[nH]1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.39
ADORA3 P0DMS8 3/20 0.39
ADORA2A P29274 2/20 0.39
DDAH1 O94760 1/20 0.33
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12877465 0.75 TGFBR1 (0.42) ADORA1GAA
SCHEMBL15134752 0.75 NISCH (0.41) HTT
SCHEMBL4336235 0.71 POLB (0.44) ADORA1ADORA3ADORA2AGAA
SCHEMBL11325781 0.71
SCHEMBL6124953 0.71
SCHEMBL13762102 0.71
SCHEMBL13668681 0.71
SCHEMBL3304072 0.67 ADORA3 (0.38) ADORA1ADORA3ADORA2A
SCHEMBL12899384 0.64 ADORA1 (0.35) ADORA1ADORA3ADORA2ADDAH1
SCHEMBL11337622 0.64 ADORA3 (0.31) ADORA1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220251042-A1 TOTAL SYNTHESIS OF PIRFENIDONE Suzhou Fude Zhaofeng Biochemical Technology Co., Ltd (CN) 2022-08-11 US disclosed
WO-2022052391-A1 METHOD FOR SYNTHESIZING VORTIOXETINE 苏州富德兆丰生化科技有限公司 2022-03-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220251042-A1 TOTAL SYNTHESIS OF PIRFENIDONE PIR, CYP2B6, CYP26B1 ADORA1 3383/4885ADORA3 3294/4885ADORA2A 3452/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.