SCHEMBL24319816

SCHEMBL24319816

C=C(CCC)c1cnc2[nH]ccc2c1C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.43
PRKCI P41743 1/20 0.43
NUDT1 P36639 1/20 0.42
JAK1 P23458 13/20 0.38
JAK3 P52333 11/20 0.38
JAK2 O60674 8/20 0.37
TTBK1 Q5TCY1 1/20 0.35
TTBK2 Q6IQ55 1/20 0.35
AURKA O14965 1/20 0.34
PRKCA P17252 1/20 0.34
KDR P35968 1/20 0.34
RPS6KA3 P51812 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21207663 0.82 NUDT1 (0.48) AXLPRKCINUDT1JAK1JAK3
SCHEMBL6128699 0.79 PRKCI (0.45) AXLPRKCINUDT1JAK1JAK3
SCHEMBL21207531 0.76 JAK1 (0.55) JAK1JAK3JAK2
SCHEMBL1082037 0.75 AXL (0.47) AXLPRKCINUDT1JAK1JAK3
SCHEMBL21207566 0.75 JAK1 (0.54) JAK1JAK3JAK2
SCHEMBL21207563 0.74 JAK3 (0.53) JAK1JAK3JAK2
SCHEMBL24495812 0.74 JAK2 (0.53) AXLPRKCINUDT1JAK1JAK3
SCHEMBL2632955 0.73 NUDT1 (0.50) AXLPRKCINUDT1JAK1JAK3
SCHEMBL31403755 0.73 NUDT1 (0.50) AXLPRKCINUDT1JAK1JAK3
SCHEMBL21207599 0.72 JAK2 (0.33) AXLPRKCINUDT1JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022067106-A1 CRYSTALLINE POLYMORPH FORM A OF A JAK INHIBITOR AND METHODS FOR ITS PREPARATION ACLARIS THERAPEUTICS, INC. (US) 2022-03-31 WO disclosed