SCHEMBL2432218

SCHEMBL2432218

Cc1ccc(F)cc1Nc1nc2ccc(C(C)C(=O)O)c(F)c2o1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.46
ITGA4 P13612 19/20 0.46
C1R P00736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2437908 0.92 ITGB1 (0.46) ITGB1ITGA4C1R
SCHEMBL2435428 0.90 KCNH2 (0.43) ITGB1ITGA4C1R
SCHEMBL2429568 0.82 ITGB1 (0.46) ITGB1ITGA4C1R
SCHEMBL14591735 0.81 ITGB1 (0.54) ITGB1ITGA4
SCHEMBL2430466 0.81 ITGB1 (0.45) ITGB1ITGA4
SCHEMBL2432759 0.81 ITGB1 (0.58) ITGB1ITGA4
SCHEMBL2433113 0.80 C1R (0.46) ITGB1ITGA4C1R
SCHEMBL14592211 0.77 ITGB1 (0.58) ITGB1ITGA4
SCHEMBL2434752 0.77 CXCL8 (0.44) ITGB1ITGA4C1R
SCHEMBL14591703 0.76 ITGB1 (0.46) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed