SCHEMBL2434752

SCHEMBL2434752

Cc1cccc(Cl)c1Nc1nc2ccc(C(C)C(=O)O)c(F)c2o1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 2/20 0.44
C1R P00736 3/20 0.43
PYGL P06737 5/20 0.39
PTGS2 P35354 2/20 0.37
MAOB P27338 1/20 0.36
LCK P06239 3/20 0.36
CHRNA7 P36544 1/20 0.36
GALK1 P51570 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2430157 0.82 PTGS2 (0.52) CXCL8C1RPTGS2ITGB1ITGA4
SCHEMBL2429568 0.80 ITGB1 (0.46) CXCL8C1RLCKITGB1ITGA4
SCHEMBL2435428 0.80 KCNH2 (0.43) C1RITGB1ITGA4
SCHEMBL14592204 0.78 ITGB1 (0.45) C1RPTGS2ITGB1ITGA4
SCHEMBL2433113 0.78 C1R (0.46) CXCL8C1RITGB1ITGA4
SCHEMBL2432218 0.77 ITGB1 (0.46) C1RITGB1ITGA4
SCHEMBL2437908 0.77 ITGB1 (0.46) C1RITGB1ITGA4
SCHEMBL2432119 0.69 ITGB1 (0.45) C1RPTGS2GALK1ITGB1ITGA4
SCHEMBL27578612 0.68 C1R (0.38) C1RITGB1ITGA4
SCHEMBL1679090 0.68 CXCL8 (0.56) CXCL8PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed