SCHEMBL24322334

SCHEMBL24322334

C1=C(c2ccnc3ccsc23)CCC1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
F2RL1 P55085 2/20 0.34
KDR P35968 2/20 0.34
ACVR1 Q04771 2/20 0.34
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
USP7 Q93009 1/20 0.33
PDPK1 O15530 1/20 0.33
PARP1 P09874 1/20 0.33
GRM2 Q14416 1/20 0.32
PSMB5 P28074 2/20 0.32
PDE10A Q9Y233 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24322146 0.76 KDR (0.35) F2RL1KDRACVR1CCNE1CDK2
SCHEMBL25156828 0.67 KDR (0.38) AXLMKNK1MKNK2KDRACVR1
SCHEMBL23716941 0.66 PDK1 (0.47) AXLMKNK1MKNK2ACVR1USP7
Hydrochloric Acid SCHEMBL6196269 0.65 AXL (0.42) AXLMKNK1MKNK2KDRPDPK1
Hydrochloric Acid SCHEMBL29564829 0.65 AXL (0.42) AXLMKNK1MKNK2KDRPDPK1
SCHEMBL23716942 0.65 CCNB2 (0.43) AXLMKNK1MKNK2KDRPDPK1
SCHEMBL4773518 0.64 ADORA2A (0.39) AXLMKNK1MKNK2ACVR1PDPK1
Hydrochloric Acid SCHEMBL4034216 0.63 PDPK1 (0.40) AXLMKNK1MKNK2KDRACVR1
SCHEMBL21393430 0.63 AXL (0.44) AXLMKNK1MKNK2KDRPDPK1
SCHEMBL4037241 0.63 AXL (0.44) AXLMKNK1MKNK2KDRPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
CN-116583283-A CDK inhibitors and their use as pharmaceuticals 普莱鲁德疗法有限公司 2023-08-11 CN disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
WO-2022061273-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS, INCORPORATED (US) 2022-03-24 WO disclosed
US-20220089608-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2022-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220089608-A1 CDK Inhibitors And Their Use As Pharmaceuticals CDK6, CDK1, CDK3 AXL 689/4885MKNK1 232/4885MKNK2 247/4885
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals CDK6, CDK1, CDK3 AXL 689/4885MKNK1 232/4885MKNK2 247/4885
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals CDK6, CDK1, CDK3 AXL 689/4885MKNK1 232/4885MKNK2 247/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.