SCHEMBL24327387

SCHEMBL24327387

C[C@@H](CO)Nc1n[nH]c2c(-c3cnn(C)c3)nc(-c3ccc(Cl)cc3)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.42
MAPK1 P28482 3/20 0.41
AXL P30530 4/20 0.40
TTK P33981 1/20 0.39
PIM1 P11309 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
HAT1 O14929 3/20 0.35
EP300 Q09472 3/20 0.35
NTRK1 P04629 1/20 0.35
KIT P10721 1/20 0.35
FLT3 P36888 1/20 0.35
MAP4K1 Q92918 1/20 0.35
CCNT1 O60563 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24328755 0.82 MAPK1 (0.39) AHRMAPK1AXLPIM1CNR1
SCHEMBL29738270 0.75 AHR (0.44) AHRMAPK1TTKCNR1CNR2
SCHEMBL29738275 0.75 AHR (0.44) AHRMAPK1TTKCNR1CNR2
SCHEMBL24327768 0.74 AHR (0.42) AHRMAPK1TTKCNR1CNR2
SCHEMBL24327393 0.73 AHR (0.42) AHRTTKKITSYK
SCHEMBL24327399 0.73 AHR (0.41) AHRTTKCNR1CNR2JAK2
SCHEMBL24327395 0.73 JAK2 (0.44) AHRMAPK1TTKCNR1CNR2
SCHEMBL24327333 0.73 JAK2 (0.44) AHRTTKCNR1CNR2JAK2
SCHEMBL24327328 0.73 JAK2 (0.44) AHRTTKCNR1CNR2JAK2
SCHEMBL24327400 0.73 AHR (0.41) AHRMAPK1TTKCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed