SCHEMBL24327388

SCHEMBL24327388

Cc1ccc(-c2cnc(Cl)c(-c3cnn(C)c3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 4/20 0.48
KDR P35968 2/20 0.48
EPHB4 P54760 1/20 0.47
TEK Q02763 1/20 0.47
LRRK2 Q5S007 1/20 0.45
MAPK1 P28482 2/20 0.43
CHEK1 O14757 1/20 0.42
CSF1R P07333 3/20 0.40
FGFR1 P11362 4/20 0.39
FGFR2 P21802 3/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
MET P08581 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
CCNT1 O60563 2/20 0.37
CCNB2 O95067 2/20 0.37
CCNE2 O96020 2/20 0.37
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
CCNE1 P24864 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29498936 1.00 FGFR3 (0.48) FGFR3KDREPHB4TEKLRRK2
SCHEMBL29498949 0.90 FGFR3 (0.56) FGFR3KDRMAPK1CHEK1CSF1R
SCHEMBL24327350 0.90 FGFR3 (0.56) FGFR3KDRMAPK1CHEK1CSF1R
SCHEMBL24327855 0.83 LRRK2 (0.58) FGFR3KDREPHB4TEKLRRK2
SCHEMBL24327401 0.80 LRRK2 (0.45) FGFR3KDREPHB4TEKLRRK2
SCHEMBL24539466 0.77 MAPK1 (0.41) FGFR3KDREPHB4TEKLRRK2
SCHEMBL24327827 0.77 FGFR3 (0.53) FGFR3KDRLRRK2MAPK1CSF1R
SCHEMBL29498933 0.77 KDR (0.53) FGFR3KDREPHB4TEKMAPK1
SCHEMBL24327347 0.77 KDR (0.53) FGFR3KDREPHB4TEKMAPK1
SCHEMBL25458623 0.76 KDR (0.48) FGFR3KDREPHB4TEKLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114369097-B Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2023-07-14 CN disclosed
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed
CN-114369097-A Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2022-04-19 CN disclosed