SCHEMBL24327557

SCHEMBL24327557

CC1Cc2cccc(Nc3nc(Cl)ncc3Cl)c2N1S

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNK O75909 9/20 0.38
CCND3 P30281 9/20 0.38
CDK9 P50750 9/20 0.38
CDK6 Q00534 9/20 0.38
CCNA2 P20248 9/20 0.38
CDK2 P24941 9/20 0.38
ALK Q9UM73 4/20 0.36
INSR P06213 2/20 0.34
MAP3K7 O43318 1/20 0.34
EGFR P00533 1/20 0.34
IGF1R P08069 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29661404 0.83 CDK7 (0.40) CDK9ALKINSREGFRIGF1R
SCHEMBL24327552 0.83 CDK7 (0.40) CDK9ALKINSREGFRIGF1R
SCHEMBL29661362 0.74 ULK1 (0.35) CCNKCCND3CDK9CDK6CCNA2
SCHEMBL24326962 0.74 ULK1 (0.35) CCNKCCND3CDK9CDK6CCNA2
SCHEMBL25004485 0.71 NOTUM (0.55) ALKMAP3K7EGFR
SCHEMBL30942601 0.71 CCNK (0.41) CCNKCCND3CDK9CDK6CCNA2
SCHEMBL29661342 0.71 CDK9 (0.43) CCNKCCND3CDK9CDK6CCNA2
SCHEMBL24327468 0.71 CDK9 (0.43) CCNKCCND3CDK9CDK6CCNA2
SCHEMBL30141686 0.71 CCNA2 (0.41) CCNKCCND3CDK9CDK6CCNA2
SCHEMBL25014389 0.70 CCNA2 (0.39) CCNKCCND3CDK9CDK6CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022063106-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEIGENE, LTD. (KY) 2022-03-31 WO disclosed