SCHEMBL2432847

SCHEMBL2432847

CCC(C(=O)O)c1cc(Cl)c(NC(=O)c2nccc3ccccc23)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.46
ITGA4 P13612 3/20 0.46
RAB9A P51151 2/20 0.41
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TP53 P04637 2/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 1/20 0.38
FLT3 P36888 1/20 0.38
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CCR1 P32246 1/20 0.37
HDAC3 O15379 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
NCOR2 Q9Y618 2/20 0.37
S1PR1 P21453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2433943 0.81 MAPT (0.48) ITGB1ITGA4MAPTTP53SMN1; SMN2
SCHEMBL2432642 0.81 EPHB3 (0.54) ITGB1ITGA4FLT3
SCHEMBL91533 0.81 ITGB1 (0.47) ITGB1ITGA4RAB9AMAPTMEN1
SCHEMBL2433516 0.80 KDM4E (0.45) TSHRALDH1A1KDM4EHDAC3HDAC1
SCHEMBL2440170 0.79 ITGB1 (0.58) ITGB1ITGA4RAB9AMAPTMEN1
SCHEMBL27581128 0.79 ITGB1 (0.46) ITGB1ITGA4RAB9AMAPTMEN1
SCHEMBL14591890 0.79 ITGB1 (0.54) ITGB1ITGA4RAB9AMAPTMEN1
SCHEMBL14626747 0.79 ITGB1 (0.55) ITGB1ITGA4RAB9AMAPTMEN1
SCHEMBL2435623 0.77 NR1I2 (0.40) RAB9AKMT2ATP53ALDH1A1SMN1; SMN2
SCHEMBL14491705 0.77 ITGB1 (0.55) ITGB1ITGA4RAB9AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed