SCHEMBL24329238

SCHEMBL24329238

Fc1cc(I)ccc1COc1cccc(C2CCNCC2)n1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 17/20 0.43
KCNH2 Q12809 1/20 0.43
HTR6 P50406 1/20 0.43
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29555248 1.00 GLP1R (0.43) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL24485665 0.89 HTR6 (0.54) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL30149360 0.89 HTR6 (0.54) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL24485288 0.87 GLP1R (0.43) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL20267985 0.87 GLP1R (0.55) GLP1RKCNH2
SCHEMBL30149289 0.87 GLP1R (0.43) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL30951873 0.87 GLP1R (0.43) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL24321924 0.87 HTR6 (0.47) GLP1RKCNH2HTR6SLC6A2SLC6A4
SCHEMBL29394844 0.87 GLP1R (0.55) GLP1RKCNH2
Hydrochloric Acid SCHEMBL25286836 0.86 GLP1R (0.54) GLP1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4227299-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF Hangzhou Zhongmeihuadong Pharmaceutical Co., Ltd. (CN) 2023-08-16 EP disclosed
EP-4227299-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF Hangzhou Zhongmeihuadong Pharmaceutical Co., Ltd. (CN) 2023-08-16 EP disclosed
CN-116348464-A Benzimidazolone GLP-1 receptor agonists and uses thereof 杭州中美华东制药有限公司 2023-06-27 CN disclosed
WO-2022078152-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF 杭州中美华东制药有限公司 2022-04-21 WO disclosed