SCHEMBL24329534

SCHEMBL24329534

CON(C)C(=O)c1cccc(COc2cccc(C3CCN(C(=O)OC(C)(C)C)CC3)n2)c1F

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 7/20 0.49
GLP1R P43220 7/20 0.43
TRPV3 Q8NET8 1/20 0.41
PRMT5 O14744 2/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24329294 0.89 TRPV3 (0.45) GPR119GLP1RTRPV3PRMT5MAPT
SCHEMBL24329295 0.89 GLP1R (0.49) GLP1RTRPV3PRMT5MAPTSMN1; SMN2
SCHEMBL24329269 0.89 GLP1R (0.47) GPR119GLP1RTRPV3PRMT5MAPT
SCHEMBL24329805 0.88 GPR119 (0.48) GPR119GLP1RTRPV3
SCHEMBL24330292 0.88 GPR119 (0.48) GPR119GLP1RTRPV3
SCHEMBL24329267 0.86 GLP1R (0.48) GPR119GLP1R
SCHEMBL29554818 0.86 GPR119 (0.48) GPR119GLP1RTRPV3
SCHEMBL29555062 0.86 GLP1R (0.48) GPR119GLP1R
SCHEMBL24329524 0.86 GPR119 (0.48) GPR119GLP1RTRPV3
SCHEMBL25340508 0.86 GPR119 (0.55) GPR119GLP1RTRPV3PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4227299-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF Hangzhou Zhongmeihuadong Pharmaceutical Co., Ltd. (CN) 2023-08-16 EP disclosed
WO-2022078152-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF 杭州中美华东制药有限公司 2022-04-21 WO disclosed