SCHEMBL2433332

SCHEMBL2433332

CCC(C(=O)O)c1cc(F)c2nc(Nc3cc(F)ccc3C)oc2c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.39
AKR1C2 P52895 6/20 0.39
AKR1B10 O60218 1/20 0.37
AKR1C4 P17516 1/20 0.37
AKR1C1 Q04828 1/20 0.37
ITGB1 P05556 7/20 0.37
ITGA4 P13612 7/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
PKM P14618 1/20 0.35
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KIT P10721 1/20 0.34
DDR2 Q16832 1/20 0.34
P2RX7 Q99572 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2433971 0.81 ITGA4 (0.43) ITGB1ITGA4P2RX7
SCHEMBL14591878 0.78 ITGA4 (0.40) ITGB1ITGA4SMN1; SMN2P2RX7
SCHEMBL14592222 0.77 ITGB1 (0.42) ITGB1ITGA4MAPTP2RX7
SCHEMBL2430466 0.74 ITGB1 (0.45) AKR1C3AKR1C2ITGB1ITGA4NPC1
SCHEMBL14591756 0.71 ITGB1 (0.39) ITGB1ITGA4P2RX7
SCHEMBL2432317 0.69 ITGA4 (0.57) ITGB1ITGA4
SCHEMBL14591744 0.69 ITGB1 (0.42) ITGB1ITGA4NPC1RAB9ASMN1; SMN2
SCHEMBL14591877 0.67 NPC1 (0.42) ITGB1ITGA4NPC1RAB9ASMN1; SMN2
SCHEMBL14591708 0.67 ITGA4 (0.53) ITGB1ITGA4
SCHEMBL2432218 0.66 ITGB1 (0.46) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed