SCHEMBL2433464

SCHEMBL2433464

CC(C(=O)O)c1ccc2nc(-c3cccnc3)oc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.60
ALDH1A1 P00352 8/20 0.60
HSD17B10 Q99714 7/20 0.60
NPC1 O15118 6/20 0.60
RAB9A P51151 6/20 0.60
HPGD P15428 5/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
TP53 P04637 3/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2C19 P33261 2/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
AKR1C3 P42330 1/20 0.57
AKR1C2 P52895 1/20 0.57
MAOA P21397 1/20 0.54
ADRA1A P35348 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
TSHR P16473 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11176670 0.80 MAOA (0.82) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL1675472 0.79 HDAC6 (0.65) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL9706321 0.78 MAOA (0.79) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL14591812 0.77 KDM4E (0.62) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL2434363 0.76 KDM4E (0.82) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL8051382 0.76 KDM4E (0.70) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL30402334 0.76 KDM4E (0.70) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL14626645 0.75 KDM4E (0.66) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL27596627 0.75 KDM4E (0.62) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL11178446 0.75 MAOA (0.55) KDM4EALDH1A1HSD17B10NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed