SCHEMBL24338908

SCHEMBL24338908

COC(=O)Cc1cc2c(CO)cccn2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.41
TSHR P16473 2/20 0.41
MAPT P10636 1/20 0.41
EGFR P00533 1/20 0.39
KDM4E B2RXH2 6/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
BAZ2B Q9UIF8 2/20 0.34
BAZ2A Q9UIF9 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
USP2 O75604 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24338940 0.87 CYP4F2 (0.45) HPGDMAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL24338066 0.83 PTGS2 (0.37) HPGDMAPTKDM4EALDH1A1BAZ2B
SCHEMBL3217965 0.78 PDE4B (0.34) TSHRMAPTALDH1A1KMT2ABAZ2B
SCHEMBL544288 0.73 KDM4E (0.41) HPGDTSHRKDM4EALDH1A1KMT2A
SCHEMBL1665456 0.73 APOBEC3A (0.46) MAPTKDM4EALDH1A1BAZ2BBAZ2A
SCHEMBL3459890 0.72 ADORA3 (0.48) MAPTKDM4EKMT2ACYP4F2CYP4A11
SCHEMBL24338568 0.72 SMN1; SMN2 (0.37) HPGDEGFRKDM4EALDH1A1SMN1; SMN2
SCHEMBL29491521 0.72 SMN1; SMN2 (0.37) HPGDTSHRMAPTKDM4EALDH1A1
SCHEMBL2961579 0.71 PDE4B (0.36) HPGDTSHRMAPTEGFRKDM4E
SCHEMBL684345 0.69 KDM4E (0.51) HPGDTSHRMAPTEGFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022068772-A1 BENZIMIDAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2022-04-07 WO disclosed