SCHEMBL2434934

SCHEMBL2434934

CC(C(=O)O)c1ccc2nc(-c3cccc4ccccc34)oc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.60
ESR2 Q92731 7/20 0.60
AKR1C3 P42330 3/20 0.57
AKR1C2 P52895 3/20 0.57
AKR1B1 P15121 1/20 0.49
MAOA P21397 1/20 0.48
ADRA1A P35348 1/20 0.48
MAPT P10636 6/20 0.48
ALDH1A1 P00352 4/20 0.48
HPGD P15428 4/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HSD17B10 Q99714 2/20 0.48
TP53 P04637 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
KDM4E B2RXH2 3/20 0.42
GAA P10253 2/20 0.42
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11178446 0.85 MAOA (0.55) AKR1C3AKR1C2MAOAADRA1AMAPT
SCHEMBL2432940 0.83 AKR1B1 (0.46) ESR1ESR2AKR1C3AKR1C2AKR1B1
SCHEMBL2433361 0.78 ITGB1 (0.47) ESR1ESR2AKR1C3AKR1C2AKR1B1
SCHEMBL2434406 0.76 ESR1 (0.63) ESR1ESR2AKR1B1MAPTALDH1A1
SCHEMBL6311736 0.76 ESR1 (1.00) ESR1ESR2MAPTALDH1A1HPGD
SCHEMBL11695908 0.75 AKR1C3 (0.59) AKR1C3AKR1C2MAOAADRA1AMAPT
SCHEMBL11697899 0.75 MAOA (0.58) ESR1ESR2AKR1C3AKR1C2MAOA
SCHEMBL27578687 0.75 ESR1 (0.62) ESR1ESR2MAPTALDH1A1HPGD
SCHEMBL25028054 0.75 ESR1 (0.72) ESR1ESR2MAPTALDH1A1HPGD
SCHEMBL11176670 0.75 MAOA (0.82) ESR1ESR2MAOAADRA1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed