SCHEMBL2432940

SCHEMBL2432940

CC(C(=O)O)c1ccc2nc(-c3nccc4ccccc34)oc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.46
MAOA P21397 1/20 0.46
ADRA1A P35348 1/20 0.46
KDM4E B2RXH2 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
GPR55 Q9Y2T6 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
AKR1C3 P42330 4/20 0.43
AKR1C2 P52895 4/20 0.43
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2434934 0.83 ESR1 (0.60) AKR1B1MAOAADRA1AKDM4ENPC1
SCHEMBL2434007 0.78 NPC1 (0.44) AKR1B1KDM4ENPC1RAB9AGPR55
SCHEMBL2429608 0.78 ITGB1 (0.55) AKR1B1KDM4ENPC1RAB9AGPR55
SCHEMBL27578581 0.77 CD74 (0.50) KDM4ENPC1RAB9AGPR55L3MBTL1
SCHEMBL11178446 0.75 MAOA (0.55) MAOAADRA1AKDM4ENPC1RAB9A
SCHEMBL2433361 0.75 ITGB1 (0.47) AKR1B1MAOAADRA1AKDM4EAKR1C3
SCHEMBL28749560 0.74 MAPT (0.48) KDM4ENPC1RAB9AGPR55L3MBTL1
SCHEMBL14592405 0.74 ITGB1 (0.52) KDM4ENPC1RAB9AGPR55L3MBTL1
SCHEMBL2433464 0.74 KDM4E (0.60) MAOAADRA1AKDM4ENPC1RAB9A
SCHEMBL28061939 0.74 NPC1 (0.56) KDM4ENPC1RAB9AGPR55L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed