SCHEMBL2435828

SCHEMBL2435828

CC(C(=O)O)c1ccc2nc(-c3cn(C)c4ccc(Cl)cc34)oc2c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.53
ADRA1A P35348 1/20 0.53
ITGB1 P05556 1/20 0.48
ITGA4 P13612 1/20 0.48
KMT2A Q03164 2/20 0.43
PTGS2 P35354 6/20 0.42
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
MEN1 O00255 1/20 0.41
ABCC4 O15439 1/20 0.41
C5 P01031 1/20 0.41
MAPT P10636 1/20 0.41
PTGS1 P23219 1/20 0.41
PDE4D Q08499 1/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2430981 0.88 ITGB1 (0.49) MAOAADRA1AITGB1ITGA4MET
SCHEMBL2435546 0.83 ITGB1 (0.48) MAOAADRA1AITGB1ITGA4MET
SCHEMBL2429639 0.82 ITGB1 (0.59) ITGB1ITGA4KMT2AMAPTMET
SCHEMBL2433361 0.80 ITGB1 (0.47) MAOAADRA1AITGB1ITGA4ABCC4
SCHEMBL11176670 0.78 MAOA (0.82) MAOAADRA1AKMT2AMEN1MAPT
SCHEMBL11178446 0.76 MAOA (0.55) MAOAADRA1APTGS2MAPT
SCHEMBL2433627 0.73 MAOA (0.48) MAOAADRA1APTGS2MAPTPTGS1
SCHEMBL2434934 0.73 ESR1 (0.60) MAOAADRA1AKMT2AMEN1MAPT
SCHEMBL2437936 0.71 ITGB1 (0.49) ITGB1ITGA4MET
SCHEMBL11637637 0.71 MAOA (0.56) MAOAADRA1AKMT2APTGS2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed