SCHEMBL2436288

SCHEMBL2436288

CC(C)(C)OC(=O)Nc1cn(-c2ccccc2)nc1NC(=O)c1ccc(CN(Cc2cccnc2)C(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.49
NAMPT P43490 2/20 0.45
HTT P42858 1/20 0.42
HDAC3 O15379 3/20 0.41
HDAC2 Q92769 3/20 0.41
NCOR2 Q9Y618 2/20 0.41
ADORA3 P0DMS8 4/20 0.41
HIF1A Q16665 1/20 0.41
EPAS1 Q99814 1/20 0.41
ALKBH5 Q6P6C2 1/20 0.40
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HDAC4 P56524 2/20 0.39
HDAC7 Q8WUI4 2/20 0.39
HDAC10 Q969S8 2/20 0.39
HDAC11 Q96DB2 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC9 Q9UKV0 2/20 0.39
HDAC5 Q9UQL6 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2438296 0.93 HDAC1 (0.46) HDAC1NAMPTHDAC3HDAC2NCOR2
SCHEMBL2435576 0.82 HDAC1 (0.60) HDAC1NAMPTHDAC3HDAC2NCOR2
SCHEMBL8235738 0.82 KDM4E (0.43) HDAC1NAMPTADORA3ALDH1A1ADORA1
SCHEMBL3765663 0.82 HDAC1 (0.49) HDAC1NAMPTHTTHDAC3HDAC2
SCHEMBL3649530 0.81 HDAC1 (0.53) HDAC1NAMPTHDAC3HDAC2NCOR2
SCHEMBL4457846 0.80 HDAC1 (0.48) HDAC1NAMPTADORA3HDAC10HDAC6
SCHEMBL2436833 0.80 ADORA3 (0.39) HDAC1NAMPTHDAC3HDAC2NCOR2
SCHEMBL2438671 0.77 HDAC1 (0.54) HDAC1NAMPTHTTHDAC3HDAC2
SCHEMBL2436494 0.77 HDAC1 (0.52) HDAC1HTTHDAC3HDAC2ADORA3
SCHEMBL2435416 0.77 HDAC1 (0.54) HDAC1HTTHDAC3HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8026260-B2 Histone deacetylase inhibitors with aryl-pyrazolyl-motifs MERCK SHARP & DOHME CORP. (US) 2011-09-27 US disclosed