SCHEMBL24363479

SCHEMBL24363479

CNc1ncnc(N)c1-c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BTK Q06187 18/20 0.53
KCNH2 Q12809 5/20 0.53
EGFR P00533 4/20 0.53
NUDT5 Q9UKK9 3/20 0.48
TEC P42680 1/20 0.48
BMX P51813 1/20 0.48
CD69 Q07108 1/20 0.48
ITK Q08881 1/20 0.48
ERBB4 Q15303 1/20 0.48
GP6 Q9HCN6 1/20 0.48
NUDT14 O95848 2/20 0.48
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CB P42338 1/20 0.47
PIK3CG P48736 1/20 0.47
PRKDC P78527 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14241118 0.85 NUDT14 (0.56) BTKKCNH2EGFRNUDT5NUDT14
SCHEMBL24363242 0.84 LCK (0.49) BTKKCNH2EGFR
SCHEMBL24363263 0.83 TTBK1 (0.52) BTKKCNH2EGFR
SCHEMBL24363230 0.79 BTK (0.69) BTKKCNH2EGFRNUDT5TEC
SCHEMBL24363496 0.78 BTK (0.68) BTKKCNH2EGFRNUDT5TEC
SCHEMBL14165704 0.77 BTK (0.70) BTKKCNH2EGFRNUDT5TEC
SCHEMBL20480850 0.77 BTK (0.70) BTKKCNH2EGFRNUDT5TEC
SCHEMBL14165691 0.77 BTK (0.70) BTKKCNH2EGFRNUDT5TEC
SCHEMBL18788360 0.77 BTK (0.48) BTKKCNH2EGFRNUDT5TEC
SCHEMBL14165430 0.76 BTK (0.66) BTKKCNH2EGFRNUDT5TEC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2718270-B1 COMPOSITIONS AND METHODS FOR THE PRODUCTION OF PYRIMIDINE AND PYRIDINE COMPOUNDS WITH BTK INHIBITORY ACTIVITY MERCK PATENT GMBH (DE) 2022-04-27 EP disclosed