SCHEMBL24370189

SCHEMBL24370189

Cc1cnc2[nH]cc(C(F)(F)F)c2n1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
MAP3K12 Q12852 6/20 0.34
MAPK1 P28482 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 1/20 0.34
HSP90AB1 P08238 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK4 Q16654 1/20 0.33
DLK1 P80370 1/20 0.32
JAK2 O60674 2/20 0.32
JAK1 P23458 2/20 0.32
JAK3 P52333 2/20 0.32
ULK1 O75385 2/20 0.32
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22201885 0.84 SYK (0.39) SYKIRAK4MAPK1HPGDPDK2
SCHEMBL25839068 0.80 MAPK1 (0.33) SYKIRAK4MAP3K12MAPK1HSP90AB1
SCHEMBL25851514 0.77 MAPK1 (0.37) SYKIRAK4MAP3K12MAPK1HPGD
SCHEMBL7950769 0.76 MAPK1 (0.39) SYKMAPK1HPGDPDK2PDK4
SCHEMBL13199608 0.73 JAK2 (0.40) SYKMAPK1HPGDHSP90AB1PDK2
SCHEMBL16946856 0.73 MAPK1 (0.37) SYKMAPK1HPGDPDK2PDK4
SCHEMBL14616216 0.73 MAPK1 (0.62) SYKMAPK1HPGDPDK2PDK4
SCHEMBL7454972 0.72 HSD17B10 (0.35) MAPK1HPGDHSD17B10ALDH1A1
SCHEMBL25839070 0.70 SYK (0.37) SYKMAPK1JAK2JAK1JAK3
SCHEMBL12253392 0.69 MAPK1 (0.36) SYKMAPK1HPGDHSD17B10PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022087634-A1 CTPS1 INHIBITORS AND USES THEREOF NIMBUS CLOTHO, INC. (US) 2022-04-28 WO disclosed