SCHEMBL24376943

SCHEMBL24376943

CCC(=O)c1ccc(Oc2ccc(C)cc2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
POLB P06746 1/20 0.50
KMT2A Q03164 2/20 0.48
LMNA P02545 2/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 1/20 0.48
CHRNA7 P36544 1/20 0.47
MEN1 O00255 1/20 0.46
CHEK2 O96017 1/20 0.46
P2RX3 P56373 3/20 0.45
MAPT P10636 1/20 0.45
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
HRH3 Q9Y5N1 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9607407 0.87 HRH3 (0.58) KDM4EKMT2ALMNAALDH1A1SMN1; SMN2
SCHEMBL14240948 0.87 HRH3 (0.56) SMN1; SMN2MAPTOPRM1OPRD1OPRK1
SCHEMBL19362950 0.84 PDE4B (0.58) KDM4ENPC1RAB9APOLBKMT2A
SCHEMBL9607063 0.83 LMNA (0.53) KDM4ELMNAMAPTOPRM1OPRD1
SCHEMBL29593315 0.83 KDM4E (0.56) KDM4ENPC1RAB9APOLBKMT2A
SCHEMBL19778853 0.83 KDM4E (0.56) KDM4ENPC1RAB9APOLBKMT2A
SCHEMBL21628634 0.83 MAPT (0.57) KDM4ENPC1RAB9APOLBKMT2A
SCHEMBL13043807 0.82 NNMT (0.61) KDM4ENPC1RAB9APOLBKMT2A
SCHEMBL6177649 0.81 KDM4E (0.55) KDM4ENPC1RAB9APOLBKMT2A
SCHEMBL21656526 0.81 LMNA (0.63) KDM4ENPC1RAB9APOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484882-B1 ISO-CITRATE DEHYDROGENASE (IDH) INHIBITOR ZHEJIANG METON PHARMACEUTICAL CO LTD (CN) 2022-04-27 EP disclosed