SCHEMBL24378068

SCHEMBL24378068

COCc1[nH]nc(CO)c1Br

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.33
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19635451 0.87 HCAR2 (0.32) HCAR2
SCHEMBL19615315 0.78 HCAR2 (0.35) HCAR2
SCHEMBL15229798 0.76 PDE4D (0.32) HCAR2
SCHEMBL19635091 0.72 PTPN1 (0.31)
SCHEMBL24378111 0.72 HCAR2 (0.30) HCAR2
SCHEMBL13683076 0.71
SCHEMBL3146744 0.69 HCAR2 (0.32) HCAR2
SCHEMBL8943452 0.64 KCNH2 (0.37) HCAR2
SCHEMBL19634996 0.64
SCHEMBL19635109 0.64 TSHR (0.44) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed