SCHEMBL24378147

SCHEMBL24378147

N=C(CCl)N1CC(C(N)=O)Oc2cc(-c3ccccc3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 14/20 0.48
SIRT3 Q9NTG7 1/20 0.41
SIRT2 Q8IXJ6 10/20 0.40
DGAT1 O75907 3/20 0.40
SOAT2 O75908 2/20 0.40
CYP2C9 P11712 1/20 0.40
SOAT1 P35610 1/20 0.40
DGAT2 Q96PD7 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24377969 0.89 SIRT1 (0.50) SIRT1SIRT3SIRT2DGAT1SOAT2
SCHEMBL24378019 0.81 SIRT1 (0.48) SIRT1SIRT3SIRT2POLB
SCHEMBL26938751 0.79 DGAT1 (0.40) SIRT1DGAT1SOAT2CYP2C9SOAT1
SCHEMBL24378125 0.73 SIRT1 (0.65) SIRT1SIRT3SIRT2TDP1
SCHEMBL26938829 0.73 SIRT1 (0.65) SIRT1SIRT3SIRT2TDP1
SCHEMBL24378118 0.73 SIRT1 (0.65) SIRT1SIRT3SIRT2TDP1
SCHEMBL24377995 0.71 SIRT1 (0.43) SIRT1SIRT3SIRT2TDP1POLB
SCHEMBL24378120 0.71 SIRT1 (0.47) SIRT1SIRT3SIRT2TDP1
SCHEMBL26938749 0.70 POLB (0.44) SIRT1CYP2C9POLB
SCHEMBL24377971 0.68 SIRT1 (0.43) SIRT1SIRT3SIRT2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022087433-A1 COVALENT INHIBITORS OF CREATINE KINASE (CK) AND USES THEREOF FOR TREATING AND PREVENTING CANCER DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-04-28 WO disclosed