SCHEMBL24399774

SCHEMBL24399774

Cc1ccc2c(Nc3cccc(Cl)c3F)ncnc2c1N

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.51
CSF1R P07333 1/20 0.51
ARAF P10398 1/20 0.51
BRAF P15056 1/20 0.51
DDR1 Q08345 1/20 0.51
DDR2 Q16832 1/20 0.51
EGFR P00533 13/20 0.50
GRM4 Q14833 1/20 0.43
TTBK1 Q5TCY1 1/20 0.41
TTBK2 Q6IQ55 1/20 0.41
EPHA2 P29317 2/20 0.41
KDR P35968 2/20 0.41
EPHB4 P54760 2/20 0.41
ERBB2 P04626 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24399558 0.82 RAF1 (0.54) RAF1CSF1RARAFBRAFDDR1
SCHEMBL30162852 0.82 RAF1 (0.54) RAF1CSF1RARAFBRAFDDR1
SCHEMBL29638701 0.77 BRAF (0.65) RAF1CSF1RARAFBRAFDDR1
SCHEMBL24399644 0.77 BRAF (0.65) RAF1CSF1RARAFBRAFDDR1
SCHEMBL6241529 0.77 EGFR (0.52) EGFRGRM4TTBK1TTBK2
SCHEMBL31406750 0.75 JAK2 (0.53) RAF1CSF1RBRAFDDR1DDR2
SCHEMBL16016709 0.74 EGFR (0.67) EGFREPHA2KDREPHB4ERBB2
SCHEMBL4737922 0.74 TTBK1 (0.75) BRAFEGFRTTBK1TTBK2
SCHEMBL26449347 0.73 EGFR (0.64) EGFREPHA2KDREPHB4ERBB2
SCHEMBL2700855 0.73 EGFR (0.64) EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230312556-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2023-10-05 US disclosed
US-20230312556-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2023-10-05 US disclosed
US-20230312556-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2023-10-05 US disclosed
EP-4238967-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2023-09-06 EP disclosed
EP-4238967-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2023-09-06 EP disclosed
WO-2022089219-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2022-05-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230312556-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF AHR, ARNT, NOTUM RAF1 2075/4885CSF1R 987/4885ARAF 553/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.