SCHEMBL24401049

SCHEMBL24401049

Cc1ncc(NC(=O)c2ccc3c(c2)OC(F)(F)O3)cc1-c1cc(F)nc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TAS2R8 Q9NYW2 1/20 0.49
RAF1 P04049 17/20 0.45
BRAF P15056 8/20 0.45
LCK P06239 2/20 0.45
KDR P35968 2/20 0.45
MAPK14 Q16539 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29747359 1.00 TAS2R8 (0.49) TAS2R8RAF1BRAFLCKKDR
SCHEMBL24401050 0.87 RAF1 (0.63) RAF1BRAF
SCHEMBL24401048 0.78 RAF1 (0.63) RAF1BRAF
SCHEMBL24401210 0.75 RAF1 (0.59) RAF1BRAF
SCHEMBL24401077 0.73 RAF1 (0.47) RAF1BRAF
SCHEMBL2951528 0.69 LCK (0.56) TAS2R8BRAFLCKKDRMAPK14
SCHEMBL30376331 0.68 SMYD3 (0.57) TAS2R8
SCHEMBL31120905 0.66 KCNQ3 (0.52)
SCHEMBL31095836 0.66 LRRK2 (0.65)
SCHEMBL1649415 0.66 TAS2R8 (1.00) TAS2R8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220135539-A1 BIARYL AMIDE COMPOUNDS, PREPARATION METHODS AND MEDICAL APPLICATIONS THEREOF Eternity Bioscience Inc. 2022-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220135539-A1 BIARYL AMIDE COMPOUNDS, PREPARATION METHODS AND MEDICAL APPLICATIONS THEREOF BRAF, NRAS, RAF1 TAS2R8 4621/4885RAF1 3/4885BRAF 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.