SCHEMBL24420243

SCHEMBL24420243

CN(Cc1ccccc1NC(=O)CC1CCCCC1)C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.51
P2RX7 Q99572 2/20 0.48
AAK1 Q2M2I8 1/20 0.47
NPC1 O15118 6/20 0.45
RAB9A P51151 5/20 0.45
TDP1 Q9NUW8 3/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 1/20 0.43
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687682 0.78 EPHX2 (0.60) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL4687186 0.77 EPHX2 (0.58) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL4690268 0.76 EPHX2 (0.57) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL4688109 0.76 EPHX2 (0.57) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL7159830 0.75 P2RX7 (0.74) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL4686987 0.75 EPHX2 (0.56) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL4688016 0.75 EPHX2 (0.56) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL4692647 0.72 EPHX2 (0.63) EPHX2P2RX7AAK1NPC1RAB9A
SCHEMBL7923968 0.71 ALDH1A1 (0.61) TDP1ALDH1A1SMN1; SMN2KMT2AKDM4E
SCHEMBL23004908 0.69 ALDH1A1 (0.44) EPHX2NPC1RAB9ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022099011-A1 BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF CYTOKINETICS, INC. (US) 2022-05-12 WO disclosed