SCHEMBL2442435

SCHEMBL2442435

CC(C)(C)OC(=O)N1CC2CCC[C@@H]2C1CNC(=O)c1nsc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.40
ACKR3 P25106 1/20 0.40
TP53 P04637 3/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL496214 1.00 HCRTR1 (0.40) HCRTR1ACKR3TP53LMNAKDM4E
SCHEMBL496277 0.87 TP53 (0.39) ACKR3TP53
SCHEMBL3641229 0.84 ACKR3 (0.40) HCRTR1ACKR3KDM4EPKM
SCHEMBL496412 0.83 HCRTR1 (0.43) HCRTR1ACKR3KDM4EPKM
SCHEMBL2446757 0.83 HCRTR1 (0.43) HCRTR1ACKR3KDM4EPKM
SCHEMBL3677156 0.81 HCRTR1 (0.40) HCRTR1ACKR3KDM4EPKM
SCHEMBL496001 0.75 HCRTR1 (0.61) HCRTR1
SCHEMBL496187 0.74 KMT2A (0.41) ACKR3LMNAKDM4EPKM
SCHEMBL496121 0.74 HTR4 (0.48) HCRTR1
SCHEMBL2441649 0.74 HTR4 (0.48) HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164847-B1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2011-09-14 EP disclosed