SCHEMBL24427802

SCHEMBL24427802

Cc1ncc(-c2cccc(C(N)=O)c2)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.49
CCND1 P24385 1/20 0.49
CCNC P24863 1/20 0.49
CDK8 P49336 1/20 0.49
CDK7 P50613 1/20 0.49
CDK9 P50750 1/20 0.49
CCNH P51946 1/20 0.49
MNAT1 P51948 1/20 0.49
CDK6 Q00534 1/20 0.49
CYP2A6 P11509 1/20 0.49
PARP1 P09874 1/20 0.47
MAP2K4 P45985 1/20 0.47
FYN P06241 7/20 0.46
EGFR P00533 2/20 0.46
GSK3B P49841 2/20 0.45
PIM1 P11309 2/20 0.45
CDC7 O00311 1/20 0.45
PLK4 O00444 1/20 0.45
CHEK1 O14757 1/20 0.45
AURKA O14965 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7894913 0.85 PRSS1 (0.50) CYP2A6
SCHEMBL4063091 0.84 MASP2 (0.56) CCNT1CCND1CCNCCDK8CDK7
Hydrochloric Acid SCHEMBL4058021 0.82 MASP2 (0.54) CCNT1CCND1CCNCCDK8CDK7
SCHEMBL24427794 0.79 F11 (0.47) CYP2A6EGFRGSK3BINSRMAPK8
SCHEMBL24427731 0.76 CYP2A6 (0.56) CYP2A6FYNGSK3BCDK1
SCHEMBL7981198 0.76 CYP2A6 (0.56) CYP2A6AXL
SCHEMBL19145369 0.75 PARP1 (0.58) CCNT1CCND1CCNCCDK8CDK7
SCHEMBL24427757 0.73 SCN2A (0.64) CYP2A6
SCHEMBL15145570 0.73 CYP2A6 (0.56) CYP2A6GSK3B
SCHEMBL24427570 0.73 CYP2A6 (0.56) CYP2A6PIM1HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3998263-A1 TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jemincare Pharmaceuticals Co., Ltd. (CN) 2022-05-18 EP disclosed