SCHEMBL24439595

SCHEMBL24439595

Cc1nc(-c2sccc2CO)cnc1OC1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 2/20 0.36
PLK1 P53350 1/20 0.36
NEK1 Q96PY6 1/20 0.36
LRRK2 Q5S007 3/20 0.34
HRH4 Q9H3N8 1/20 0.33
RIPK1 Q13546 1/20 0.33
HDAC3 O15379 3/20 0.32
CDK9 P50750 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
FFAR4 Q5NUL3 1/20 0.32
CNR1 P21554 1/20 0.32
CDK4 P11802 1/20 0.32
HDAC1 Q13547 2/20 0.32
CDK2 P24941 1/20 0.31
KDR P35968 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
ABCB11 O95342 1/20 0.31
SLCO1B1 Q9Y6L6 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29601754 1.00 NEK2 (0.36) NEK2PLK1NEK1LRRK2HRH4
SCHEMBL28756107 0.85 SLCO1B1 (0.47) NEK2PLK1NEK1FFAR4ABCB11
SCHEMBL29602427 0.83 CNR1 (0.33) LRRK2HDAC3CDK9HDAC6FFAR4
SCHEMBL24439682 0.83 CNR1 (0.33) LRRK2HDAC3CDK9HDAC6FFAR4
SCHEMBL29517393 0.83 SLCO1B1 (0.40) NEK2PLK1NEK1FFAR4ABCB11
SCHEMBL24439594 0.83 SLCO1B1 (0.40) NEK2PLK1NEK1FFAR4ABCB11
SCHEMBL24439314 0.82 LPAR1 (0.33) RIPK1ABCB11SLCO1B1
SCHEMBL29672126 0.82 LPAR1 (0.33) RIPK1ABCB11SLCO1B1
SCHEMBL24439775 0.81 FFAR4 (0.34) NEK2LRRK2HRH4HDAC3CDK9
SCHEMBL29602253 0.81 FFAR4 (0.34) NEK2LRRK2HRH4HDAC3CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100625-A1 NITROGEN-SUBSTITUTED AMINOCARBONATE THIOPHENE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed