SCHEMBL24439682

SCHEMBL24439682

Cc1nc(-c2sc(Cl)cc2CO)cnc1OC1CCCCC1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.33
FFAR4 Q5NUL3 3/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
LRRK2 Q5S007 2/20 0.33
LIMK1 P53667 1/20 0.32
LIMK2 P53671 1/20 0.32
HDAC3 O15379 3/20 0.32
CDK9 P50750 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
HDAC1 Q13547 2/20 0.32
PDGFRB P09619 2/20 0.31
PDGFRA P16234 2/20 0.31
CDK4 P11802 1/20 0.31
GRM5 P41594 1/20 0.30
ABCB11 O95342 1/20 0.30
SLCO1B1 Q9Y6L6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29602427 1.00 CNR1 (0.33) CNR1FFAR4S1PR1S1PR3LRRK2
SCHEMBL24441641 0.89 LOX (0.34) FFAR4LRRK2LIMK1LIMK2HDAC3
SCHEMBL28755958 0.85 SLCO1B1 (0.46) FFAR4ABCB11SLCO1B1
SCHEMBL29577386 0.84 ABCB11 (0.38) CNR1FFAR4S1PR1S1PR3ABCB11
SCHEMBL24439681 0.84 ABCB11 (0.38) CNR1FFAR4S1PR1S1PR3ABCB11
SCHEMBL24439595 0.83 NEK2 (0.36) CNR1FFAR4LRRK2HDAC3CDK9
SCHEMBL29601754 0.83 NEK2 (0.36) CNR1FFAR4LRRK2HDAC3CDK9
SCHEMBL24439734 0.83 KMO (0.36)
SCHEMBL29672295 0.83 KMO (0.36)
SCHEMBL24439741 0.81 SLCO1B1 (0.39) FFAR4S1PR1S1PR3ABCB11SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100625-A1 NITROGEN-SUBSTITUTED AMINOCARBONATE THIOPHENE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed