SCHEMBL24439737

SCHEMBL24439737

COC(=O)[C@H]1CCC[C@H](Oc2ncc(-c3sccc3C=O)nc2C)C1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.38
SLCO1B1 Q9Y6L6 1/20 0.38
KMT2A Q03164 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
NEK2 P51955 3/20 0.32
LPAR1 Q92633 1/20 0.31
PLK1 P53350 1/20 0.31
NEK1 Q96PY6 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
IRAK1 P51617 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29517766 1.00 ABCB11 (0.38) ABCB11SLCO1B1KMT2AFFAR4NEK2
SCHEMBL28755991 0.91 SLCO1B1 (0.46) ABCB11SLCO1B1FFAR4NEK2LPAR1
SCHEMBL29517393 0.87 SLCO1B1 (0.40) ABCB11SLCO1B1KMT2AFFAR4NEK2
SCHEMBL24439594 0.87 SLCO1B1 (0.40) ABCB11SLCO1B1KMT2AFFAR4NEK2
SCHEMBL24440689 0.86 LPAR1 (0.41) ABCB11SLCO1B1KMT2ALPAR1ALDH1A1
SCHEMBL24439775 0.84 FFAR4 (0.34) ABCB11SLCO1B1FFAR4NEK2EGFR
SCHEMBL29602253 0.84 FFAR4 (0.34) ABCB11SLCO1B1FFAR4NEK2EGFR
SCHEMBL24441487 0.84 ABCB11 (0.37) ABCB11SLCO1B1FFAR4
SCHEMBL29576270 0.84 ABCB11 (0.37) ABCB11SLCO1B1FFAR4
SCHEMBL24439357 0.83 KMT2A (0.35) ABCB11SLCO1B1KMT2ALPAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100625-A1 NITROGEN-SUBSTITUTED AMINOCARBONATE THIOPHENE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
CN-114456147-A Oxygen substituted amino carbonate thiophene compounds 武汉人福创新药物研发中心有限公司 2022-05-10 CN disclosed