SCHEMBL24449337

SCHEMBL24449337

Cc1cc(-n2nc(C#N)c(=O)[nH]c2=O)cc(C)c1Oc1c[nH]c(=O)c(C(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB P10828 19/20 0.56
THRA P10827 17/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C8 P10632 1/20 0.56
UGT1A1 P22309 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24449974 0.89 THRB (0.55) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL28656735 0.89 THRB (0.55) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL24408097 0.89 THRA (0.70) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL24449978 0.85 THRA (0.63) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL31347914 0.85 THRA (0.63) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL24407902 0.85 THRB (0.54) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL24449961 0.84 THRB (0.51) THRBTHRACYP2C9CYP2C8UGT1A1
SCHEMBL22632645 0.83 THRB (0.49) THRBTHRACYP2C9CYP2C8
SCHEMBL29414670 0.83 THRB (0.49) THRBTHRACYP2C9CYP2C8
SCHEMBL24449962 0.83 THRB (0.51) THRBTHRACYP2C9CYP2C8UGT1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12338206-B2 Compounds and their uses as thyroid hormone receptor agonists NANJING RUIJIE PHARMA CO., LTD. (CN) 2025-06-24 US disclosed
CN-119431265-A Compound as thyroid hormone receptor agonist 南京瑞捷医药科技有限公司 2025-02-14 CN disclosed
CN-113474335-B Compounds and their use as thyroid hormone receptor agonists 南京瑞捷医药科技有限公司 2024-12-03 CN disclosed
EP-4240730-A1 2-PYRIDONES AS THYROID HORMONE RECEPTOR MODULATORS Aligos Therapeutics, Inc. (US) 2023-09-13 EP disclosed
CN-116710443-A 2-pyridones as thyroid hormone receptor modulators 阿利戈斯治疗公司 2023-09-05 CN disclosed
US-20220162161-A1 Novel compounds and their uses as thyroid hormone receptor agonists NANJING RUIJIE PHARMA CO., LTD. (CN) 2022-05-26 US disclosed
WO-2022099044-A1 2-PYRIDONES AS THYROID HORMONE RECEPTOR MODULATORS ALIGOS THERAPEUTICS, INC. (US) 2022-05-12 WO disclosed
CN-113474335-A Novel compounds and their use as thyroid hormone receptor agonists 南京瑞捷医药科技有限公司 2021-10-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220162161-A1 Novel compounds and their uses as thyroid hormone receptor agonists THRA, THRB, TSHR THRB 2/4885THRA 1/4885CYP2C9 1825/4885
US-12338206-B2 Compounds and their uses as thyroid hormone receptor agonists THRA, THRB, TSHR THRB 2/4885THRA 1/4885CYP2C9 1854/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.