SCHEMBL2445209

SCHEMBL2445209

O=C(CBr)Nc1nc(-c2cc(F)c(OCC3CC3)c(Cl)c2)cs1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 2/20 0.50
TRPA1 O75762 3/20 0.48
ABL1 P00519 5/20 0.44
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
WNT3A P56704 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2445205 0.96 FFAR4 (0.47) FFAR4TRPA1ABL1RAB9ANPC1
SCHEMBL481106 0.93 TRPA1 (0.45) FFAR4TRPA1RAB9ANPC1MEN1
SCHEMBL2447447 0.93 ABL1 (0.47) FFAR4TRPA1ABL1RAB9ANPC1
SCHEMBL480890 0.89 ABL1 (0.46) TRPA1ABL1RAB9ANPC1MEN1
SCHEMBL480419 0.89 FFAR4 (0.48) FFAR4TRPA1RAB9ANPC1MEN1
SCHEMBL4408309 0.89 ABL1 (0.45) TRPA1ABL1RAB9ANPC1KMT2A
SCHEMBL15580544 0.86 TRPA1 (0.50) TRPA1ABL1RAB9AMEN1KMT2A
SCHEMBL2440259 0.85 TRPA1 (0.49) TRPA1ABL1RAB9AMEN1KMT2A
SCHEMBL480355 0.85 TRPA1 (0.60) TRPA1ABL1RAB9AMEN1KMT2A
SCHEMBL480700 0.84 TRPA1 (0.55) TRPA1ABL1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed