SCHEMBL2447447

SCHEMBL2447447

O=C(CBr)Nc1nc(-c2cc(Cl)c(OCC3CC3)c(Cl)c2)cs1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.47
TRPA1 O75762 5/20 0.44
CLK1 P49759 1/20 0.43
MAPT P10636 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480890 0.96 ABL1 (0.46) ABL1TRPA1CLK1MAPTPI4KB
SCHEMBL4408309 0.95 ABL1 (0.45) ABL1TRPA1CLK1MAPTPI4KB
SCHEMBL2445209 0.93 FFAR4 (0.50) ABL1TRPA1FFAR4MEN1NPC1
SCHEMBL2445205 0.90 FFAR4 (0.47) ABL1TRPA1FFAR4MEN1NPC1
SCHEMBL481106 0.88 TRPA1 (0.45) TRPA1FFAR4MEN1NPC1RAB9A
SCHEMBL2443035 0.85 MAPT (0.49) ABL1TRPA1CLK1MAPTPI4KB
SCHEMBL480419 0.84 FFAR4 (0.48) TRPA1FFAR4MEN1NPC1RAB9A
SCHEMBL2450413 0.83 ABL1 (0.51) ABL1TRPA1CLK1MAPTMEN1
SCHEMBL2450859 0.83 TRPA1 (0.48) ABL1TRPA1CLK1MAPTPI4KB
SCHEMBL480411 0.82 TRPA1 (0.58) ABL1TRPA1CLK1MAPTPI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed