SCHEMBL24464244

SCHEMBL24464244

Cc1cn(C2CC2)nc(C)c1=O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 12/20 0.37
TLR7 Q9NYK1 4/20 0.37
TLR9 Q9NR96 3/20 0.37
TLR4 O00206 2/20 0.37
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
DRD3 P35462 2/20 0.35
PDE10A Q9Y233 1/20 0.34
AADAT Q8N5Z0 1/20 0.33
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB2 P47870 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21258472 0.84 DRD2 (0.39) TLR8TLR7TLR9TLR4DRD2
SCHEMBL24152761 0.76 ALDH1A1 (0.39) TLR8TLR7TLR9TLR4DRD2
SCHEMBL25712191 0.76 SMYD3 (0.37) DRD2DRD4DRD3AADATPDE4D
SCHEMBL26298923 0.76 LRRK2 (0.41) DRD2DRD4DRD3GABRA1GABRB2
SCHEMBL25718397 0.76 SMYD3 (0.37) DRD2DRD4DRD3AADATPDE4D
SCHEMBL23584944 0.75 DRD2 (0.44) TLR8TLR7TLR9TLR4DRD2
SCHEMBL22258794 0.74 ALDH1A1 (0.41) DRD2DRD4DRD3AADATALDH1A1
SCHEMBL23584998 0.73 DRD2 (0.42) TLR8TLR7TLR9TLR4DRD2
SCHEMBL20689124 0.72 KDM5A (0.42) DRD2DRD4DRD3GABRA1GABRB2
SCHEMBL21863534 0.72 DRD2 (0.37) DRD2DRD4DRD3AADATGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4005637-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2022-06-01 EP disclosed