SCHEMBL24467263

SCHEMBL24467263

COc1cc(C)c(Sc2cnc(Nc3ccc(CN(C)C)cn3)s2)cc1C

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 13/20 0.66
BTK Q06187 12/20 0.48
TXK P42681 10/20 0.48
ITK Q08881 8/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23365933 0.81 JAK3 (1.00) JAK3BTKTXKITK
SCHEMBL20162010 0.80 JAK3 (0.63) JAK3BTKTXKITK
SCHEMBL24467190 0.77 BTK (0.71) JAK3BTKTXKITK
SCHEMBL24467251 0.75 JAK3 (0.46) JAK3BTKTXKITK
SCHEMBL24467153 0.71 JAK3 (0.48) JAK3BTKTXKITK
SCHEMBL24467287 0.69 JAK3 (0.69) JAK3BTKTXKITK
SCHEMBL20162005 0.68 JAK3 (0.39) JAK3BTKTXKITK
SCHEMBL24467248 0.68 ITK (0.70) JAK3BTKTXKITK
SCHEMBL24467347 0.67 JAK3 (0.68) JAK3BTKTXKITK
SCHEMBL24467232 0.65 BTK (0.68) JAK3BTKTXKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3534899-B1 COMPOUNDS AND METHODS FOR MODULATING INTERLEUKIN-2-INDUCIBLE T-CELL KINASE CORVUS PHARMACEUTICALS INC (US) 2022-06-01 EP disclosed