SCHEMBL24474358

SCHEMBL24474358

COCOc1cccc(O)c1C(=O)/C=C/c1ccc(Br)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 8/20 0.60
NFKB2 Q00653 8/20 0.60
RELA Q04206 8/20 0.60
SLC5A1 P13866 1/20 0.50
SLC5A2 P31639 1/20 0.50
BACE1 P56817 3/20 0.49
MAOB P27338 2/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
TP53 P04637 1/20 0.47
MDM2 Q00987 1/20 0.47
MAOA P21397 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25205679 0.89 NFKB1 (0.63) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL30383093 0.89 NFKB1 (0.63) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL25205681 0.89 NFKB1 (0.63) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL25184989 0.86 AURKA (0.61) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL25265167 0.86 AURKA (0.61) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL31232999 0.86 AURKA (0.61) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL1728182 0.84 NFKB1 (0.58) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL1728183 0.84 NFKB1 (0.58) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL16098173 0.84 MAOB (0.61) NFKB1NFKB2RELABACE1MAOB
SCHEMBL16100756 0.84 MAOB (0.61) NFKB1NFKB2RELABACE1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022113047-A1 4'-SUBSTITUTED ANALOGUES OF FISETIN AND THEIR USE IN THE TREATMENT OF CANCER STELLENBOSCH UNIVERSITY (ZA) 2022-06-02 WO disclosed