SCHEMBL24477338

SCHEMBL24477338

CCC(C)c1cc(=O)n2c(n1)[nH]c1ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.46
ALDH1A1 P00352 8/20 0.46
HPGD P15428 6/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
RAB9A P51151 4/20 0.46
HSD17B10 Q99714 3/20 0.46
MAPK10 P53779 1/20 0.46
GAA P10253 5/20 0.43
GLA P06280 4/20 0.43
MAPT P10636 4/20 0.43
HTT P42858 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
LMNA P02545 3/20 0.42
PDE2A O00408 1/20 0.41
PDE6D O43924 1/20 0.41
PDE8A O60658 1/20 0.41
PDE5A O76074 1/20 0.41
PDE9A O76083 1/20 0.41
PDE8B O95263 1/20 0.41
PDE6A P16499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23295690 0.87 ALDH1A1 (0.49) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL31653998 0.79 KDM4E (0.50) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL19411063 0.76 KDM4E (0.56) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL24477383 0.76 MEN1 (0.44) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL24477316 0.76 MEN1 (0.46) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL24477314 0.76 MEN1 (0.46) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL24477317 0.76 MEN1 (0.46) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL24477339 0.76 ALDH1A1 (0.36) ALDH1A1HPGDSMN1; SMN2RAB9AHTT
SCHEMBL24477379 0.75 KDM4E (0.51) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A
SCHEMBL24477393 0.75 KDM4E (0.51) KDM4EALDH1A1HPGDSMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022111473-A1 COMPOUNDS AS MRGPRX2 ANTAGONISTS BIOARDIS LLC (US) 2022-06-02 WO disclosed
WO-2022111473-A1 COMPOUNDS AS MRGPRX2 ANTAGONISTS BIOARDIS LLC (US) 2022-06-02 WO disclosed